Publications

A synergistic inhibitor development strategy against human UDP‐galactose‐4‐epimerase

Browne William M, Pettinger Jonathan, Weckwerth Teresa, Purkiss Andrew, Lok Sing Hei, Penicaut Louisa, Ogrodowicz Roksana, Prema Raveena, Kunzelmann Simone, Roustan Chloe, Bineva‐Todd Ganka, Pieters Saskia, Zappacosta Francesca, Doherty Alfred E, Oram Isobel, Soudy Christelle, Quinlan Robert, Redmond Joanna, Kjaer Svend, House David, Mouilleron Stephane, Bush Jacob T, Schumann Benjamin

Angewandte Chemie International Edition Vol 65 (2026)

https://doi.org/10.1002/anie.202520304

Expedited SARS‐CoV‐2 main protease inhibitor discovery through modular 'direct‐to‐biology' screening

Wilders Harry, Biggs George, Rowe Sam M, Cawood Emma E, Riziotis Ioannis G, Rendina Alan R, Grant Emma K, Pettinger Jonathan, Fallon David J, Skehel Mark, House David, Tomkinson Nicholas C O, Bush Jacob T

Angewandte Chemie Vol 137 (2025)

https://doi.org/10.1002/ange.202418314

Robust proteome profiling of cysteine-reactive fragments using label-free chemoproteomics

Biggs George S, Cawood Emma E, Vuorinen Aini, McCarthy William J, Wilders Harry, Riziotis Ioannis G, van der Zouwen Antonie J, Pettinger Jonathan, Nightingale Luke, Chen Peiling, Powell Andrew J, House David, Boulton Simon J, Skehel J Mark, Rittinger Katrin, Bush Jacob T

Nature Communications Vol 16, pp. 73 (2025)

https://doi.org/10.1038/s41467-024-55057-5

Photoaffinity labelling displacement assay using multiple recombinant protein domains

Fallon David J, Phillipou Alex, Schofield Christopher J, House David, Tomkinson Nicholas C O, Bush Jacob T

Biochemical Journal Vol 480, pp. 1183-1197 (2023)

https://doi.org/10.1042/bcj20230129

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